Dominique Schols

Publications

• Optimization of Triazolo[4,5-d]pyrimidines Towards Human CC Chemokine Receptor 7 (CCR7) Antagonists
  European Journal of Medicinal Chemistry. Mar, 2023  |   Pubmed ID: 36924670
• A Regioselective Step-by-step CCl Functionalization Approach Affords a Novel Family of CArTh'Th''H Fullerene Derivatives with Promising Antiviral Properties
  Chemical Communications (Cambridge, England). Mar, 2023  |   Pubmed ID: 36916636
• Exploration of Pyrido[3,4-]pyrimidines As Antagonists of the Human Chemokine Receptor CXCR2
  Molecules (Basel, Switzerland). Feb, 2023  |   Pubmed ID: 36903345
• Visible-Light-Promoted Tandem Thiol-Ene Click Reaction/Transannular Cyclization and Regioselective Cyclopropane Ring-Opening to Construct Sulfur-Containing Diterpenes
  Organic Letters. Feb, 2023  |   Pubmed ID: 36662155
• FLUIDOT: A Modular Microfluidic Platform for Single-Cell Study and Retrieval, with Applications in Drug Tolerance Screening and Antibody Mining
  Small Methods. Mar, 2023  |   Pubmed ID: 36642827
• Design and Synthesis of a New Series of Hybrids of Functionalised N-[(1H-1,2,3-triazol-4-yl)methyl]quinazoline-2,4-dione with Antiviral Activity Against Respiratory Syncytial Virus
  Antiviral Research. Jan, 2023  |   Pubmed ID: 36587900
• Development of a Live Biotherapeutic Throat Spray with Lactobacilli Targeting Respiratory Viral Infections
  Microbial Biotechnology. Jan, 2023  |   Pubmed ID: 36468246
• Identification of Polyphenol Derivatives As Novel SARS-CoV-2 and DENV Non-Nucleoside RdRp Inhibitors
  Molecules (Basel, Switzerland). Dec, 2022  |   Pubmed ID: 36615354
• Systemic Cytokines and GlycA Discriminate Disease Status and Predict Corticosteroid Response in HTLV-1-associated Neuroinflammation
  Journal of Neuroinflammation. Dec, 2022  |   Pubmed ID: 36482436
• Synthesis and Evaluation of 3-alkynyl-5-aryl-7-aza-indoles As Broad-spectrum Antiviral Agents
  Frontiers in Chemistry. 2022  |   Pubmed ID: 36385995
• A Stabilized CXCL9(74-103)-derived Peptide Selectively Inhibits Proliferation, Adhesion and Metastasis of Tumor Cells That Express High Levels of Heparan Sulfate
  International Journal of Biological Macromolecules. Dec, 2022  |   Pubmed ID: 36272565
• Design, Synthesis, Anti-Varicella-Zoster and Antimicrobial Activity of (Isoxazolidin-3-yl)Phosphonate Conjugates of N1-Functionalised Quinazoline-2,4-Diones
  Molecules (Basel, Switzerland). Oct, 2022  |   Pubmed ID: 36235061
• Can We Attenuate Ischaemia-reperfusion Injury of Allografts in a Porcine Left Lung Transplant Models by Adsorption of Cytokines?
  European Journal of Cardio-thoracic Surgery : Official Journal of the European Association for Cardio-thoracic Surgery. Dec, 2022  |   Pubmed ID: 36214633
• Corrigendum: Innate Lymphoid Cells Are Required to Induce Airway Hyperreactivity in a Murine Neutrophilic Asthma Model
  Frontiers in Immunology. 2022  |   Pubmed ID: 36211405
• Carbohydrate-binding Protein from Stinging Nettle As Fusion Inhibitor for SARS-CoV-2 Variants of Concern
  Frontiers in Cellular and Infection Microbiology. 2022  |   Pubmed ID: 36111239
• Triphosphate Prodrugs of the Anti-HIV-Active Compound 3'-Deoxy-3'-fluorothymidine (FLT)
  Journal of Medicinal Chemistry. Sep, 2022  |   Pubmed ID: 36099330
• Cellular Electrical Impedance As a Method to Decipher CCR7 Signalling and Biased Agonism
  International Journal of Molecular Sciences. Aug, 2022  |   Pubmed ID: 36012168
• Cryo-EM Structures of Wild-type and E138K/M184I Mutant HIV-1 RT/DNA Complexed with Inhibitors Doravirine and Rilpivirine
  Proceedings of the National Academy of Sciences of the United States of America. Jul, 2022  |   Pubmed ID: 35858448
• Potent Neutralizing Anti-SARS-CoV-2 Human Antibodies Cure Infection with SARS-CoV-2 Variants in Hamster Model
  IScience. Aug, 2022  |   Pubmed ID: 35813873
• SARS-CoV-2 Virion Infectivity and Cytokine Production in Primary Human Airway Epithelial Cells
  Viruses. May, 2022  |   Pubmed ID: 35632693
• The Discovery of Zika Virus NS2B-NS3 Inhibitors with Antiviral Activity Via an Integrated Virtual Screening Approach
  European Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences. Aug, 2022  |   Pubmed ID: 35618201
• Discovery of 2-Phenylquinolines with Broad-Spectrum Anti-coronavirus Activity
  ACS Medicinal Chemistry Letters. May, 2022  |   Pubmed ID: 35571875
• Stimulation of the Atypical Chemokine Receptor 3 (ACKR3) by a Small-molecule Agonist Attenuates Fibrosis in a Preclinical Liver but Not Lung Injury Model
  Cellular and Molecular Life Sciences : CMLS. May, 2022  |   Pubmed ID: 35562519
• Effect of Particle Carriers for Intraperitoneal Drug Delivery on the Course of Ovarian Cancer and Its Immune Microenvironment in a Mouse Model
  Pharmaceutics. Mar, 2022  |   Pubmed ID: 35456521
• In Silico Design, Synthesis and Anti-HIV Activity of Quinoline Derivatives As Non-nucleoside Reverse Transcriptase Inhibitors (NNRTIs)
  Computational Biology and Chemistry. Jun, 2022  |   Pubmed ID: 35395595
• Innate Lymphoid Cells Are Required to Induce Airway Hyperreactivity in a Murine Neutrophilic Asthma Model
  Frontiers in Immunology. 2022  |   Pubmed ID: 35371094
• A Set of Experimentally Validated Decoys for the Human CC Chemokine Receptor 7 (CCR7) Obtained by Virtual Screening
  Frontiers in Pharmacology. 2022  |   Pubmed ID: 35370691
• Identification of Novel Chemotypes As CXCR2 Antagonists Via a Scaffold Hopping Approach from a Thiazolo[4,5-d]pyrimidine
  European Journal of Medicinal Chemistry. May, 2022  |   Pubmed ID: 35313168
• Circulating Donor-Specific Anti-HLA Antibodies Associate With Immune Activation Independent of Kidney Transplant Histopathological Findings
  Frontiers in Immunology. 2022  |   Pubmed ID: 35281018
• Targeting Chemokine Receptors from the Inside-out: Discovery and Development of Small-molecule Intracellular Antagonists
  Chemical Communications (Cambridge, England). Mar, 2022  |   Pubmed ID: 35274633
• Synthesis, in Vitro Cytotoxicity, molecular Docking and ADME Study of Some Indolin-2-one Linked 1,2,3-triazole Derivatives
  Computational Biology and Chemistry. Apr, 2022  |   Pubmed ID: 35168158
• Anthranilamides with Quinoline and β-carboline Scaffolds: Design, Synthesis, and Biological Activity
  Molecular Diversity. Oct, 2022  |   Pubmed ID: 34997441
• Atypical Response to Bacterial Coinfection and Persistent Neutrophilic Bronchoalveolar Inflammation Distinguish Critical COVID-19 from Influenza
  JCI Insight. Jan, 2022  |   Pubmed ID: 34793331
• Lung Microenvironments and Disease Progression in Fibrotic Hypersensitivity Pneumonitis
  American Journal of Respiratory and Critical Care Medicine. Jan, 2022  |   Pubmed ID: 34724391
• Discovery of ( ±)-3-(1H-pyrazol-1-yl)-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4] Thiadiazine Derivatives with Promising in Vitro Anticoronavirus and Antitumoral Activity
  Molecular Diversity. Jun, 2022  |   Pubmed ID: 34165689
• Itaconic Acid Hybrids As Potential Anticancer Agents
  Molecular Diversity. Feb, 2022  |   Pubmed ID: 33043404
• Deciphering the Role of Extracellular Vesicles Derived from ZIKV-Infected HcMEC/D3 Cells on the Blood-Brain Barrier System
  Viruses. Nov, 2021  |   Pubmed ID: 34960632
• Sliding of HIV-1 Reverse Transcriptase over DNA Creates a Transient P Pocket - Targeting P-pocket by Fragment Screening
  Nature Communications. Dec, 2021  |   Pubmed ID: 34880240
• Skeleton Binding Protein-1-mediated Parasite Sequestration Inhibits Spontaneous Resolution of Malaria-associated Acute Respiratory Distress Syndrome
  PLoS Pathogens. Nov, 2021  |   Pubmed ID: 34843584
• Peripherally-driven Myeloid NFkB and IFN/ISG Responses Predict Malignancy Risk, Survival, and Immunotherapy Regime in Ovarian Cancer
  Journal for Immunotherapy of Cancer. Nov, 2021  |   Pubmed ID: 34795003
• Synthesis and Anti-HIV Activity of a Novel Series of Isoquinoline-Based CXCR4 Antagonists
  Molecules (Basel, Switzerland). Oct, 2021  |   Pubmed ID: 34684878
• D-Peptide-Based Probe for CXCR4-Targeted Molecular Imaging and Radionuclide Therapy
  Pharmaceutics. Oct, 2021  |   Pubmed ID: 34683912
• A Proteomic Study on the Membrane Protein Fraction of T Cells Confirms High Substrate Selectivity for the ER Translocation Inhibitor Cyclotriazadisulfonamide
  Molecular & Cellular Proteomics : MCP. 2021  |   Pubmed ID: 34481949
• Water-Promoted Reaction of CArCl Compounds with Thiophenes Delivers a Family of Multifunctional Fullerene Derivatives with Selective Antiviral Properties
  Organic Letters. Sep, 2021  |   Pubmed ID: 34468156
• Exploring the DNTP -binding Site of HIV-1 Reverse Transcriptase for Inhibitor Design
  European Journal of Medicinal Chemistry. Dec, 2021  |   Pubmed ID: 34425311
• Novel N-Substituted 3-Aryl-4-(diethoxyphosphoryl)azetidin-2-ones As Antibiotic Enhancers and Antiviral Agents in Search for a Successful Treatment of Complex Infections
  International Journal of Molecular Sciences. Jul, 2021  |   Pubmed ID: 34360797
• Internal Disulfide Bonding and Glycosylation of Interleukin-7 Protect Against Proteolytic Inactivation by Neutrophil Metalloproteinases and Serine Proteases
  Frontiers in Immunology. 2021  |   Pubmed ID: 34276694
• Labyrinthopeptin A1 Inhibits Dengue and Zika Virus Infection by Interfering with the Viral Phospholipid Membrane
  Virology. Oct, 2021  |   Pubmed ID: 34274562
• Broad Spectrum Anti-coronavirus Activity of a Series of Anti-malaria Quinoline Analogues
  Antiviral Research. Sep, 2021  |   Pubmed ID: 34217752
• Active Components from Prevent HIV-1 Entry by Distinct Mechanisms of Action
  International Journal of Molecular Sciences. May, 2021  |   Pubmed ID: 34068829
• A Novel Series of Indole Alkaloid Derivatives Inhibit Dengue and Zika Virus Infection by Interference with the Viral Replication Complex
  Antimicrobial Agents and Chemotherapy. Jul, 2021  |   Pubmed ID: 34001508
• Small Molecule Cyclotriazadisulfonamide Abrogates the Upregulation of the Human Receptors CD4 and 4-1BB and Suppresses In Vitro Activation and Proliferation of T Lymphocytes
  Frontiers in Immunology. 2021  |   Pubmed ID: 33968048
• Biological Characterization of Ligands Targeting the Human CC Chemokine Receptor 8 (CCR8) Reveals the Biased Signaling Properties of Small Molecule Agonists
  Biochemical Pharmacology. Jun, 2021  |   Pubmed ID: 33872569
• Corrigendum to 'Discovery of HIV Entry Inhibitors Via a Hybrid CXCR4 and CCR5 Receptor Pharmacophore-based Virtual Screening Approach' [European Journal of Pharmaceutical Sciences 155 (2020) 105537]
  European Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences. Jul, 2021  |   Pubmed ID: 33814256
• FO-SPR Biosensor Calibrated with Recombinant Extracellular Vesicles Enables Specific and Sensitive Detection Directly in Complex Matrices
  Journal of Extracellular Vesicles. Feb, 2021  |   Pubmed ID: 33664936
• Synthesis, in Silico ADME, Molecular Docking and in Vitro Cytotoxicity Evaluation of Stilbene Linked 1,2,3-triazoles
  Heliyon. Jan, 2021  |   Pubmed ID: 33553718
• A Novel Experimental Porcine Model to Assess the Impact of Differential Pulmonary Blood Flow on Ischemia-reperfusion Injury After Unilateral Lung Transplantation
  Intensive Care Medicine Experimental. Feb, 2021  |   Pubmed ID: 33543363
• Discovery of 3-phenyl- and 3-N-piperidinyl-isothiazolo[4,3-b]pyridines As Highly Potent Inhibitors of Cyclin G-associated Kinase
  European Journal of Medicinal Chemistry. Mar, 2021  |   Pubmed ID: 33497888
• Palladium-catalyzed Cross-coupling Reactions on a Bromo-naphthalene Scaffold in the Search for Novel Human CC Chemokine Receptor 8 (CCR8) Antagonists
  Bioorganic Chemistry. Feb, 2021  |   Pubmed ID: 33383325
• Characterization of the Carbohydrate-Binding Agents HHA, GNA, and UDA As Inhibitors of Influenza A and B Virus Replication
  Antimicrobial Agents and Chemotherapy. Feb, 2021  |   Pubmed ID: 33288640
• Synthesis, Molecular Docking and Preliminary Antileukemic Activity of 4-Methoxybenzyl Derivatives Bearing Imidazo[2,1-b][1,3,4]thiadiazole
  Chemistry & Biodiversity. Feb, 2021  |   Pubmed ID: 33274824
• A Single-dose Live-attenuated YF17D-vectored SARS-CoV-2 Vaccine Candidate
  Nature. 02, 2021  |   Pubmed ID: 33260195
• γ-Non-Symmetrically Dimasked TriPPPro Prodrugs As Potential Antiviral Agents Against HIV
  ChemMedChem. Feb, 2021  |   Pubmed ID: 33089929
• STAT2 Signaling Restricts Viral Dissemination but Drives Severe Pneumonia in SARS-CoV-2 Infected Hamsters
  Nature Communications. 11, 2020  |   Pubmed ID: 33203860
• γ-Ketobenzyl-Modified Nucleoside Triphosphate Prodrugs As Potential Antivirals
  Journal of Medicinal Chemistry. Nov, 2020  |   Pubmed ID: 33186038
• Development of a Novel SPR Assay to Study CXCR4-Ligand Interactions
  Biosensors. Oct, 2020  |   Pubmed ID: 33096938
• Thiophene-based Water-soluble Fullerene Derivatives As Highly Potent Antiherpetic Pharmaceuticals
  Organic & Biomolecular Chemistry. Nov, 2020  |   Pubmed ID: 33084716
• Alkylated Benzimidazoles: Design, Synthesis, Docking, DFT Analysis, ADMET Property, Molecular Dynamics and Activity Against HIV and YFV
  Computational Biology and Chemistry. Dec, 2020  |   Pubmed ID: 33068917
• Membrane Permeable, Bioreversibly Modified Prodrugs of Nucleoside Diphosphate-γ-Phosphonates
  Journal of Medicinal Chemistry. Oct, 2020  |   Pubmed ID: 32991174
• Synthesis of New Riboflavin Modified ODNs: Effect of Riboflavin Moiety on the G-quadruplex Arrangement and Stability
  Bioorganic Chemistry. Nov, 2020  |   Pubmed ID: 32919132
• Discovery of HIV Entry Inhibitors Via a Hybrid CXCR4 and CCR5 Receptor Pharmacophore-based Virtual Screening Approach
  European Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences. Dec, 2020  |   Pubmed ID: 32890663
• Water-soluble Fullerene-based Nanostructures with Promising Antiviral and Myogenic Activity
  Chemical Communications (Cambridge, England). Sep, 2020  |   Pubmed ID: 32748905
• Lipophilic Triphosphate Prodrugs of Various Nucleoside Analogues
  Journal of Medicinal Chemistry. Jul, 2020  |   Pubmed ID: 32515595
• Anti-HIV-Active Nucleoside Triphosphate Prodrugs
  Journal of Medicinal Chemistry. Jun, 2020  |   Pubmed ID: 32421343
• Prodrugs of γ-Alkyl-Modified Nucleoside Triphosphates: Improved Inhibition of HIV Reverse Transcriptase
  Angewandte Chemie (International Ed. in English). Dec, 2020  |   Pubmed ID: 32379948
• Early Protein Expression Profile in Bronchoalveolar Lavage Fluid and Clinical Outcomes in Primary Graft Dysfunction After Lung Transplantation
  European Journal of Cardio-thoracic Surgery : Official Journal of the European Association for Cardio-thoracic Surgery. Aug, 2020  |   Pubmed ID: 32267918
• A Chimeric Yellow Fever-Zika Virus Vaccine Candidate Fully Protects Against Yellow Fever Virus Infection in Mice
  Emerging Microbes & Infections. 2020  |   Pubmed ID: 32116148
• Design, Synthesis and Biological Evaluation of 2-alkoxycarbonyl-3-anilinoindoles As a New Class of Potent Inhibitors of Tubulin Polymerization
  Bioorganic Chemistry. Apr, 2020  |   Pubmed ID: 32086053
• Tryptophan Trimers and Tetramers Inhibit Dengue and Zika Virus Replication by Interfering with Viral Attachment Processes
  Antimicrobial Agents and Chemotherapy. Feb, 2020  |   Pubmed ID: 31932383
• Preprotein Signature for Full Susceptibility to the Co-translational Translocation Inhibitor Cyclotriazadisulfonamide
  Traffic (Copenhagen, Denmark). Feb, 2020  |   Pubmed ID: 31675144
• Design, Synthesis and Antiviral Evaluation of Novel Acyclic Phosphonate Nucleotide Analogs with Triazolo[4,5-]pyridine, Imidazo[4,5-]pyridine and Imidazo[4,5-]pyridin-2(3)-one Systems
  Nucleosides, Nucleotides & Nucleic Acids. 2020  |   Pubmed ID: 31550993
• Cu PET Imaging of the CXCR4 Chemokine Receptor Using a Cross-Bridged Cyclam Bis-Tetraazamacrocyclic Antagonist
  Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. Jan, 2020  |   Pubmed ID: 31201250
• Design, Synthesis, and Biological Evaluation of Novel C5-Modified Pyrimidine Ribofuranonucleosides As Potential Antitumor Or/and Antiviral Agents
  Medicinal Chemistry (Shariqah (United Arab Emirates)). 2020  |   Pubmed ID: 30799795
• Acyclic Nucleoside Phosphonates Containing the Amide Bond: Hydroxy Derivatives
  Monatshefte Fur Chemie. 2019  |   Pubmed ID: 32214483
• Novel Isoxazolidine and γ-Lactam Analogues of Homonucleosides
  Molecules (Basel, Switzerland). Nov, 2019  |   Pubmed ID: 31698778
• A Unique Class of Lignin Derivatives Displays Broad Anti-HIV Activity by Interacting with the Viral Envelope
  Virus Research. Dec, 2019  |   Pubmed ID: 31618614
• Antitumor and Antiviral Activities of 4-substituted 1,2,3-triazolyl-2,3-dibenzyl-L-ascorbic Acid Derivatives
  European Journal of Medicinal Chemistry. Dec, 2019  |   Pubmed ID: 31586832
• Modifications in the Branched Arms of a Class of Dual Inhibitors of HIV and EV71 Replication Expand Their Antiviral Spectrum
  Antiviral Research. Aug, 2019  |   Pubmed ID: 31228490
• Diversion of the Arbuzov Reaction: Alkylation of C-Cl Instead of Phosphonic Ester Formation on the Fullerene Cage
  Organic & Biomolecular Chemistry. Aug, 2019  |   Pubmed ID: 31169856
• Advantages and Shortcomings of Cell-based Electrical Impedance Measurements As a GPCR Drug Discovery Tool
  Biosensors & Bioelectronics. Jul, 2019  |   Pubmed ID: 31077988
• Highly Stable Hexitol Based XNA Aptamers Targeting the Vascular Endothelial Growth Factor
  Nucleic Acids Research. Jun, 2019  |   Pubmed ID: 30968117
• Acetate As a Model for Aspartate-based CXCR4 Chemokine Receptor Binding of Cobalt and Nickel Complexes of Cross-bridged Tetraazamacrocycles
  Dalton Transactions (Cambridge, England : 2003). Feb, 2019  |   Pubmed ID: 30729243
• Synthesis and Anti-HIV Activity of Guanine Modified Fluorinated Acyclic Nucleoside Phosphonate Derivatives
  Chemistry & Biodiversity. Feb, 2019  |   Pubmed ID: 30431702
• Synthesis, Anti-Varicella-Zoster Virus and Anti-Cytomegalovirus Activity of 4,5-Disubstituted 1,2,3-(1H)-Triazoles
  Medicinal Chemistry (Shariqah (United Arab Emirates)). 2019  |   Pubmed ID: 30411688
• A Yellow Fever-Zika Chimeric Virus Vaccine Candidate Protects Against Zika Infection and Congenital Malformations in Mice
  NPJ Vaccines. 2018  |   Pubmed ID: 30564463
• CXCR4-targeting Nanobodies Differentially Inhibit CXCR4 Function and HIV Entry
  Biochemical Pharmacology. Dec, 2018  |   Pubmed ID: 30342024
• Nanobody-Fc Constructs Targeting Chemokine Receptor CXCR4 Potently Inhibit Signaling and CXCR4-mediated HIV-entry and Induce Antibody Effector Functions
  Biochemical Pharmacology. Dec, 2018  |   Pubmed ID: 30342023
• Peroxynitrite Exposure of CXCL12 Impairs Monocyte, Lymphocyte and Endothelial Cell Chemotaxis, Lymphocyte Extravasation and Anti-HIV-1 Activity
  Frontiers in Immunology. 2018  |   Pubmed ID: 30233568
• Design, Synthesis, in Vitro Antiproliferative Activity and Apoptosis-inducing Studies of 1-(3',4',5'-trimethoxyphenyl)-3-(2'-alkoxycarbonylindolyl)-2-propen-1-one Derivatives Obtained by a Molecular Hybridisation Approach
  Journal of Enzyme Inhibition and Medicinal Chemistry. Dec, 2018  |   Pubmed ID: 30141353
• Synthesis of a 3'-C-ethynyl-β-d-ribofuranose Purine Nucleoside Library: Discovery of C7-deazapurine Analogs As Potent Antiproliferative Nucleosides
  European Journal of Medicinal Chemistry. Sep, 2018  |   Pubmed ID: 30098481
• Isoxazolidine Conjugates of N3-Substituted 6-Bromoquinazolinones-Synthesis, Anti-Varizella-Zoster Virus, and Anti-Cytomegalovirus Activity
  Molecules (Basel, Switzerland). Jul, 2018  |   Pubmed ID: 30060562
• Engineering Lactobacillus Rhamnosus GG and GR-1 to Express HIV-inhibiting Griffithsin
  International Journal of Antimicrobial Agents. Nov, 2018  |   Pubmed ID: 30040991
• Asymmetric Primaquine and Halogenaniline Fumardiamides As Novel Biologically Active Michael Acceptors
  Molecules (Basel, Switzerland). Jul, 2018  |   Pubmed ID: 30011922
• Iterative Chemical Engineering of Vancomycin Leads to Novel Vancomycin Analogs With a High Therapeutic Index
  Frontiers in Microbiology. 2018  |   Pubmed ID: 29930540
• CXCR7/ACKR3-targeting Ligands Interfere with X7 HIV-1 and HIV-2 Entry and Replication in Human Host Cells
  Heliyon. Mar, 2018  |   Pubmed ID: 29560468
• Chloro-1,4-dimethyl-9H-carbazole Derivatives Displaying Anti-HIV Activity
  Molecules (Basel, Switzerland). Jan, 2018  |   Pubmed ID: 29385738
• Aminomethylation of Heliomycin: Preparation and Anticancer Characterization of the First Series of Semi-synthetic Derivatives
  European Journal of Medicinal Chemistry. Jan, 2018  |   Pubmed ID: 29137865
• Signaling Properties of the Human Chemokine Receptors CXCR4 and CXCR7 by Cellular Electric Impedance Measurements
  PloS One. 2017  |   Pubmed ID: 28945785
• Design, Synthesis, and the Biological Evaluation of a New Series of Acyclic 1,2,3-Triazole Nucleosides
  Archiv Der Pharmazie. Sep, 2017  |   Pubmed ID: 28763115
• Expanding the Antiviral Spectrum of 3-Fluoro-2-(phosphonomethoxy)propyl Acyclic Nucleoside Phosphonates: Diamyl Aspartate Amidate Prodrugs
  Journal of Medicinal Chemistry. Jul, 2017  |   Pubmed ID: 28682067
• Immunoregulatory Effects of Multipotent Adult Progenitor Cells in a Porcine Ex Vivo Lung Perfusion Model
  Stem Cell Research & Therapy. Jul, 2017  |   Pubmed ID: 28676074
• Comparison of Cell-based Assays for the Identification and Evaluation of Competitive CXCR4 Inhibitors
  PloS One. 2017  |   Pubmed ID: 28410420
• Synthesis and Ativiral Activity of 5-(Benzylthio)-4-carbamyl-1,2,3-triazoles Against Human Cytomegalovirus (CMV) and Varicella-zoster Virus (VZV)
  Medicinal Chemistry (Shariqah (United Arab Emirates)). 2017  |   Pubmed ID: 28290250
• Structure-activity Relationship Studies on a Trp Dendrimer with Dual Activities Against HIV and Enterovirus A71. Modifications on the Amino Acid
  Antiviral Research. Mar, 2017  |   Pubmed ID: 28017762
• A Proteomic Survey Indicates Sortilin As a Secondary Substrate of the ER Translocation Inhibitor Cyclotriazadisulfonamide (CADA)
  Molecular & Cellular Proteomics : MCP. Feb, 2017  |   Pubmed ID: 27998951
• Synthesis of Different Types of Alkoxy Fullerene Derivatives from Chlorofullerene CCl
  Organic & Biomolecular Chemistry. Jan, 2017  |   Pubmed ID: 27830866
• Synthesis, Anti-varicella-zoster Virus and Anti-cytomegalovirus Activity of Quinazoline-2,4-diones Containing Isoxazolidine and Phosphonate Substructures
  European Journal of Medicinal Chemistry. Jan, 2017  |   Pubmed ID: 27750154
• Novel Isoxazolidine Analogues of Homonucleosides and Homonucleotides
  Tetrahedron. Dec, 2016  |   Pubmed ID: 32287430
• Synthesis of Novel -acyl--d-glucopyranosylamines and Ureas As Potential Lead Cytostatic Agents
  Medicinal Chemistry Research : an International Journal for Rapid Communications on Design and Mechanisms of Action of Biologically Active Agents. 2016  |   Pubmed ID: 32214768
• Synthesis, Antiviral, Cytotoxic and Cytostatic Evaluation of -(phosphonoalkyl)uracil Derivatives
  Monatshefte Fur Chemie. 2016  |   Pubmed ID: 32214481
• Acyclic Nucleoside Phosphonates Containing the Amide Bond
  Monatshefte Fur Chemie. 2016  |   Pubmed ID: 27881885
• The Lectin-like Protein 1 in Lactobacillus Rhamnosus GR-1 Mediates Tissue-specific Adherence to Vaginal Epithelium and Inhibits Urogenital Pathogens
  Scientific Reports. Nov, 2016  |   Pubmed ID: 27869151
• High Mannose-specific Lectin Msl Mediates Key Interactions of the Vaginal Lactobacillus Plantarum Isolate CMPG5300
  Scientific Reports. Nov, 2016  |   Pubmed ID: 27853317
• Synthesis and the Biological Activity of Phosphonylated 1,2,3-Triazolenaphthalimide Conjugates
  Molecules (Basel, Switzerland). Oct, 2016  |   Pubmed ID: 27792200
• Lectin-Like Molecules of Lactobacillus Rhamnosus GG Inhibit Pathogenic Escherichia Coli and Salmonella Biofilm Formation
  PloS One. 2016  |   Pubmed ID: 27537843
• Aspartate-Based CXCR4 Chemokine Receptor Binding of Cross-Bridged Tetraazamacrocyclic Copper(II) and Zinc(II) Complexes
  Chemistry (Weinheim an Der Bergstrasse, Germany). Aug, 2016  |   Pubmed ID: 27458983
• New Isoxazolidine-Conjugates of Quinazolinones-Synthesis, Antiviral and Cytostatic Activity
  Molecules (Basel, Switzerland). Jul, 2016  |   Pubmed ID: 27455228
• Lectin-Glycan Interaction Network-Based Identification of Host Receptors of Microbial Pathogenic Adhesins
  MBio. 07, 2016  |   Pubmed ID: 27406561
• Synthesis of Novel Chiral Sulfonamide-Bearing 1,2,4-Triazole-3-thione Analogs Derived from D- and L-Phenylalanine Esters As Potential Anti-Influenza Agents
  Chirality. 06, 2016  |   Pubmed ID: 27225330
• The Viral Polymerase Inhibitor 7-Deaza-2'-C-Methyladenosine Is a Potent Inhibitor of In Vitro Zika Virus Replication and Delays Disease Progression in a Robust Mouse Infection Model
  PLoS Neglected Tropical Diseases. 05, 2016  |   Pubmed ID: 27163257
• Membrane-permeable Triphosphate Prodrugs of Nucleoside Analogues
  Angewandte Chemie (International Ed. in English). Apr, 2016  |   Pubmed ID: 27008042
• Tuning Side Arm Electronics in Unsymmetrical Cyclotriazadisulfonamide (CADA) Endoplasmic Reticulum (ER) Translocation Inhibitors to Improve Their Human Cluster of Differentiation 4 (CD4) Receptor Down-Modulating Potencies
  Journal of Medicinal Chemistry. Mar, 2016  |   Pubmed ID: 26974263
• Exploring the Purine Core of 3'-C-ethynyladenosine (EAdo) in Search of Novel Nucleoside Therapeutics
  Bioorganic & Medicinal Chemistry Letters. Apr, 2016  |   Pubmed ID: 26965865
• Discovery of Antitumor Anthra[2,3-b]furan-3-carboxamides: Optimization of Synthesis and Evaluation of Antitumor Properties
  European Journal of Medicinal Chemistry. Apr, 2016  |   Pubmed ID: 26890118
• Synthesis and Bioactivity of Novel Trisubstituted Triazole Nucleosides
  Nucleosides, Nucleotides & Nucleic Acids. 2016  |   Pubmed ID: 26854981
• Vascular Endothelial Growth Factor Pathway in Endometriosis: Genetic Variants and Plasma Biomarkers
  Fertility and Sterility. Apr, 2016  |   Pubmed ID: 26773192
• Design, Synthesis, and Antiviral Activity of Novel Ribonucleosides of 1,2,3-Triazolylbenzyl-aminophosphonates
  Archiv Der Pharmazie. Jan, 2016  |   Pubmed ID: 26575425
• Lipophilic Prodrugs of Nucleoside Triphosphates As Biochemical Probes and Potential Antivirals
  Nature Communications. Oct, 2015  |   Pubmed ID: 26503889
• Phosphonylated Acyclic Guanosine Analogues with the 1,2,3-Triazole Linker
  Molecules (Basel, Switzerland). Oct, 2015  |   Pubmed ID: 26501246
• BAL Neutrophilia in Azithromycin-treated Lung Transplant Recipients: Clinical Significance
  Transplant Immunology. Sep, 2015  |   Pubmed ID: 26168736
• Design, Antiviral and Cytostatic Properties of Isoxazolidine-containing Amonafide Analogues
  Bioorganic & Medicinal Chemistry. Jul, 2015  |   Pubmed ID: 26001344
• An Easy Microwave-assisted Synthesis of C8-alkynyl Adenine Pyranonucleosides As Novel Cytotoxic Antitumor Agents
  Frontiers in Chemistry. 2015  |   Pubmed ID: 25853123
• Branched-chain Sugar Nucleosides: Stereocontrolled Synthesis and Bioevaluation of Novel 3'-C-trifluoromethyl and 3'-C-methyl Pyranonucleosides
  Carbohydrate Research. Apr, 2015  |   Pubmed ID: 25812993
• NICTABA and UDA, Two GlcNAc-binding Lectins with Unique Antiviral Activity Profiles
  The Journal of Antimicrobial Chemotherapy. 2015  |   Pubmed ID: 25700718
• Differential Cytokine, Chemokine and Growth Factor Expression in Phenotypes of Chronic Lung Allograft Dysfunction
  Transplantation. Jan, 2015  |   Pubmed ID: 25050473
• Signal Peptide-binding Drug As a Selective Inhibitor of Co-translational Protein Translocation
  PLoS Biology. Dec, 2014  |   Pubmed ID: 25460167
• 2-(4-Chlorobenzyl)-6-arylimidazo[2,1-b][1,3,4]thiadiazoles: Synthesis, Cytotoxic Activity and Mechanism of Action
  European Journal of Medicinal Chemistry. Sep, 2014  |   Pubmed ID: 25064346
• Design, Synthesis, Antiviral and Cytostatic Activity of ω-(1H-1,2,3-triazol-1-yl)(polyhydroxy)alkylphosphonates As Acyclic Nucleotide Analogues
  Bioorganic & Medicinal Chemistry. Jul, 2014  |   Pubmed ID: 24906510
• Sulfated Escherichia Coli K5 Polysaccharide Derivatives Inhibit Dengue Virus Infection of Human Microvascular Endothelial Cells by Interacting with the Viral Envelope Protein E Domain III
  PloS One. 2013  |   Pubmed ID: 24015314
• A Multi-targeted Drug Candidate with Dual Anti-HIV and Anti-HSV Activity
  PLoS Pathogens. 2013  |   Pubmed ID: 23935482
• Algal Lectins As Potential HIV Microbicide Candidates
  Marine Drugs. Jul, 2012  |   Pubmed ID: 22851920
• Carbohydrate-binding Agents Efficiently Prevent Dendritic Cell-specific Intercellular Adhesion Molecule-3-grabbing Nonintegrin (DC-SIGN)-directed HIV-1 Transmission to T Lymphocytes
  Molecular Pharmacology. Jan, 2007  |   Pubmed ID: 17056872
• Mutational Pathways, Resistance Profile, and Side Effects of Cyanovirin Relative to Human Immunodeficiency Virus Type 1 Strains with N-glycan Deletions in Their Gp120 Envelopes
  Journal of Virology. Sep, 2006  |   Pubmed ID: 16912292