Dominique Schols

Laboratory of Virology and Chemotherapy, KU Leuven

Affiliated withKU Leuven

Research Area

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JoVE Journal Publications

ArticleTotal : 3	Year
Publication title Cited by 12	2018
Publication title Cited by 22	2018
Publication title Cited by 2	2023

Other Publications

Article	Year
Mutational pathways, resistance profile, and side effects of cyanovirin relative to human immunodeficiency virus type 1 strains with N-glycan deletions in their gp120 envelopes. Journal of virology\| PubMed ID: 16912292	2006
Carbohydrate-binding agents efficiently prevent dendritic cell-specific intercellular adhesion molecule-3-grabbing nonintegrin (DC-SIGN)-directed HIV-1 transmission to T lymphocytes. Molecular pharmacology\| PubMed ID: 17056872	2007
Algal lectins as potential HIV microbicide candidates. Marine drugs\| PubMed ID: 22851920	2012
A multi-targeted drug candidate with dual anti-HIV and anti-HSV activity. PLoS pathogens\| PubMed ID: 23935482	2013
Sulfated Escherichia coli K5 polysaccharide derivatives inhibit dengue virus infection of human microvascular endothelial cells by interacting with the viral envelope protein E domain III. PloS one\| PubMed ID: 24015314	2013
Design, synthesis, antiviral and cytostatic activity of ω-(1H-1,2,3-triazol-1-yl)(polyhydroxy)alkylphosphonates as acyclic nucleotide analogues. Bioorganic & medicinal chemistry\| PubMed ID: 24906510	2014
Differential cytokine, chemokine and growth factor expression in phenotypes of chronic lung allograft dysfunction. Transplantation\| PubMed ID: 25050473	2015
2-(4-Chlorobenzyl)-6-arylimidazo[2,1-b][1,3,4]thiadiazoles: synthesis, cytotoxic activity and mechanism of action. European journal of medicinal chemistry\| PubMed ID: 25064346	2014
Signal peptide-binding drug as a selective inhibitor of co-translational protein translocation. PLoS biology\| PubMed ID: 25460167	2014
NICTABA and UDA, two GlcNAc-binding lectins with unique antiviral activity profiles. The Journal of antimicrobial chemotherapy\| PubMed ID: 25700718	2015
Branched-chain sugar nucleosides: stereocontrolled synthesis and bioevaluation of novel 3'-C-trifluoromethyl and 3'-C-methyl pyranonucleosides. Carbohydrate research\| PubMed ID: 25812993	2015
An easy microwave-assisted synthesis of C8-alkynyl adenine pyranonucleosides as novel cytotoxic antitumor agents. Frontiers in chemistry\| PubMed ID: 25853123	2015
Design, antiviral and cytostatic properties of isoxazolidine-containing amonafide analogues. Bioorganic & medicinal chemistry\| PubMed ID: 26001344	2015
BAL neutrophilia in azithromycin-treated lung transplant recipients: Clinical significance. Transplant immunology\| PubMed ID: 26168736	2015
Phosphonylated Acyclic Guanosine Analogues with the 1,2,3-Triazole Linker. Molecules (Basel, Switzerland)\| PubMed ID: 26501246	2015
Lipophilic prodrugs of nucleoside triphosphates as biochemical probes and potential antivirals. Nature communications\| PubMed ID: 26503889	2015
Design, Synthesis, and Antiviral Activity of Novel Ribonucleosides of 1,2,3-Triazolylbenzyl-aminophosphonates. Archiv der Pharmazie\| PubMed ID: 26575425	2016
Vascular endothelial growth factor pathway in endometriosis: genetic variants and plasma biomarkers. Fertility and sterility\| PubMed ID: 26773192	2016
Synthesis and Bioactivity of Novel Trisubstituted Triazole Nucleosides. Nucleosides, nucleotides & nucleic acids\| PubMed ID: 26854981	2016
Discovery of antitumor anthra[2,3-b]furan-3-carboxamides: Optimization of synthesis and evaluation of antitumor properties. European journal of medicinal chemistry\| PubMed ID: 26890118	2016
Exploring the purine core of 3'-C-ethynyladenosine (EAdo) in search of novel nucleoside therapeutics. Bioorganic & medicinal chemistry letters\| PubMed ID: 26965865	2016
Tuning Side Arm Electronics in Unsymmetrical Cyclotriazadisulfonamide (CADA) Endoplasmic Reticulum (ER) Translocation Inhibitors to Improve their Human Cluster of Differentiation 4 (CD4) Rec... Journal of medicinal chemistry\| PubMed ID: 26974263	2016
Membrane-permeable Triphosphate Prodrugs of Nucleoside Analogues. Angewandte Chemie (International ed. in English)\| PubMed ID: 27008042	2016
The Viral Polymerase Inhibitor 7-Deaza-2'-C-Methyladenosine Is a Potent Inhibitor of In Vitro Zika Virus Replication and Delays Disease Progression in a Robust Mouse Infection Model. PLoS neglected tropical diseases\| PubMed ID: 27163257	2016
Synthesis of Novel Chiral Sulfonamide-Bearing 1,2,4-Triazole-3-thione Analogs Derived from D- and L-Phenylalanine Esters as Potential Anti-Influenza Agents. Chirality\| PubMed ID: 27225330	2016
Lectin-Glycan Interaction Network-Based Identification of Host Receptors of Microbial Pathogenic Adhesins. mBio\| PubMed ID: 27406561	2016
New Isoxazolidine-Conjugates of Quinazolinones-Synthesis, Antiviral and Cytostatic Activity. Molecules (Basel, Switzerland)\| PubMed ID: 27455228	2016
Aspartate-Based CXCR4 Chemokine Receptor Binding of Cross-Bridged Tetraazamacrocyclic Copper(II) and Zinc(II) Complexes. Chemistry (Weinheim an der Bergstrasse, Germany)\| PubMed ID: 27458983	2016
Lectin-Like Molecules of Lactobacillus rhamnosus GG Inhibit Pathogenic Escherichia coli and Salmonella Biofilm Formation. PloS one\| PubMed ID: 27537843	2016
Synthesis, anti-varicella-zoster virus and anti-cytomegalovirus activity of quinazoline-2,4-diones containing isoxazolidine and phosphonate substructures. European journal of medicinal chemistry\| PubMed ID: 27750154	2017
Synthesis and the Biological Activity of Phosphonylated 1,2,3-Triazolenaphthalimide Conjugates. Molecules (Basel, Switzerland)\| PubMed ID: 27792200	2016
Synthesis of different types of alkoxy fullerene derivatives from chlorofullerene CCl. Organic & biomolecular chemistry\| PubMed ID: 27830866	2017
High mannose-specific lectin Msl mediates key interactions of the vaginal Lactobacillus plantarum isolate CMPG5300. Scientific reports\| PubMed ID: 27853317	2016
The lectin-like protein 1 in Lactobacillus rhamnosus GR-1 mediates tissue-specific adherence to vaginal epithelium and inhibits urogenital pathogens. Scientific reports\| PubMed ID: 27869151	2016
Acyclic nucleoside phosphonates containing the amide bond. Monatshefte fur chemie\| PubMed ID: 27881885	2016
Structure-activity relationship studies on a Trp dendrimer with dual activities against HIV and enterovirus A71. Modifications on the amino acid. Antiviral research\| PubMed ID: 28017762	2017
Synthesis and Ativiral Activity of 5-(Benzylthio)-4-carbamyl-1,2,3-triazoles Against Human Cytomegalovirus (CMV) and Varicella-zoster Virus (VZV). Medicinal chemistry (Shariqah (United Arab Emirates))\| PubMed ID: 28290250	2017
Comparison of cell-based assays for the identification and evaluation of competitive CXCR4 inhibitors. PloS one\| PubMed ID: 28410420	2017
Immunoregulatory effects of multipotent adult progenitor cells in a porcine ex vivo lung perfusion model. Stem cell research & therapy\| PubMed ID: 28676074	2017
Expanding the Antiviral Spectrum of 3-Fluoro-2-(phosphonomethoxy)propyl Acyclic Nucleoside Phosphonates: Diamyl Aspartate Amidate Prodrugs. Journal of medicinal chemistry\| PubMed ID: 28682067	2017
Design, Synthesis, and the Biological Evaluation of a New Series of Acyclic 1,2,3-Triazole Nucleosides. Archiv der Pharmazie\| PubMed ID: 28763115	2017
Signaling properties of the human chemokine receptors CXCR4 and CXCR7 by cellular electric impedance measurements. PloS one\| PubMed ID: 28945785	2017
Aminomethylation of heliomycin: Preparation and anticancer characterization of the first series of semi-synthetic derivatives. European journal of medicinal chemistry\| PubMed ID: 29137865	2018
Chloro-1,4-dimethyl-9H-carbazole Derivatives Displaying Anti-HIV Activity. Molecules (Basel, Switzerland)\| PubMed ID: 29385738	2018
A Proteomic Survey Indicates Sortilin as a Secondary Substrate of the ER Translocation Inhibitor Cyclotriazadisulfonamide (CADA). Molecular & cellular proteomics : MCP\| PubMed ID: 27998951	2017
CXCR7/ACKR3-targeting ligands interfere with X7 HIV-1 and HIV-2 entry and replication in human host cells. Heliyon\| PubMed ID: 29560468	2018
Iterative Chemical Engineering of Vancomycin Leads to Novel Vancomycin Analogs With a High Therapeutic Index. Frontiers in microbiology\| PubMed ID: 29930540	2018
Asymmetric Primaquine and Halogenaniline Fumardiamides as Novel Biologically Active Michael Acceptors. Molecules (Basel, Switzerland)\| PubMed ID: 30011922	2018
Engineering Lactobacillus rhamnosus GG and GR-1 to express HIV-inhibiting griffithsin. International journal of antimicrobial agents\| PubMed ID: 30040991	2018
Isoxazolidine Conjugates of N3-Substituted 6-Bromoquinazolinones-Synthesis, Anti-Varizella-Zoster Virus, and Anti-Cytomegalovirus Activity. Molecules (Basel, Switzerland)\| PubMed ID: 30060562	2018
Synthesis of a 3'-C-ethynyl-β-d-ribofuranose purine nucleoside library: Discovery of C7-deazapurine analogs as potent antiproliferative nucleosides. European journal of medicinal chemistry\| PubMed ID: 30098481	2018
Design, synthesis, in vitro antiproliferative activity and apoptosis-inducing studies of 1-(3',4',5'-trimethoxyphenyl)-3-(2'-alkoxycarbonylindolyl)-2-propen-1-one derivatives obtained by a m... Journal of enzyme inhibition and medicinal chemistry\| PubMed ID: 30141353	2018
Peroxynitrite Exposure of CXCL12 Impairs Monocyte, Lymphocyte and Endothelial Cell Chemotaxis, Lymphocyte Extravasation and Anti-HIV-1 Activity. Frontiers in immunology\| PubMed ID: 30233568	2018
Nanobody-Fc constructs targeting chemokine receptor CXCR4 potently inhibit signaling and CXCR4-mediated HIV-entry and induce antibody effector functions. Biochemical pharmacology\| PubMed ID: 30342023	2018
CXCR4-targeting nanobodies differentially inhibit CXCR4 function and HIV entry. Biochemical pharmacology\| PubMed ID: 30342024	2018
Synthesis, Anti-Varicella-Zoster Virus and Anti-Cytomegalovirus Activity of 4,5-Disubstituted 1,2,3-(1H)-Triazoles. Medicinal chemistry (Shariqah (United Arab Emirates))\| PubMed ID: 30411688	2019
Synthesis and Anti-HIV Activity of Guanine Modified Fluorinated Acyclic Nucleoside Phosphonate Derivatives. Chemistry & biodiversity\| PubMed ID: 30431702	2019
A yellow fever-Zika chimeric virus vaccine candidate protects against Zika infection and congenital malformations in mice. NPJ vaccines\| PubMed ID: 30564463	2018
Acetate as a model for aspartate-based CXCR4 chemokine receptor binding of cobalt and nickel complexes of cross-bridged tetraazamacrocycles. Dalton transactions (Cambridge, England : 2003)\| PubMed ID: 30729243	2019
Design, Synthesis, and Biological Evaluation of Novel C5-Modified Pyrimidine Ribofuranonucleosides as Potential Antitumor or/and Antiviral Agents. Medicinal chemistry (Shariqah (United Arab Emirates))\| PubMed ID: 30799795	2020
Highly stable hexitol based XNA aptamers targeting the vascular endothelial growth factor. Nucleic acids research\| PubMed ID: 30968117	2019
Advantages and shortcomings of cell-based electrical impedance measurements as a GPCR drug discovery tool. Biosensors & bioelectronics\| PubMed ID: 31077988	2019
Diversion of the Arbuzov reaction: alkylation of C-Cl instead of phosphonic ester formation on the fullerene cage. Organic & biomolecular chemistry\| PubMed ID: 31169856	2019
Cu PET Imaging of the CXCR4 Chemokine Receptor Using a Cross-Bridged Cyclam Bis-Tetraazamacrocyclic Antagonist. Journal of nuclear medicine : official publication, Society of Nuclear Medicine\| PubMed ID: 31201250	2020
Modifications in the branched arms of a class of dual inhibitors of HIV and EV71 replication expand their antiviral spectrum. Antiviral research\| PubMed ID: 31228490	2019
Design, synthesis and antiviral evaluation of novel acyclic phosphonate nucleotide analogs with triazolo[4,5-]pyridine, imidazo[4,5-]pyridine and imidazo[4,5-]pyridin-2(3)-one systems. Nucleosides, nucleotides & nucleic acids\| PubMed ID: 31550993	2020
Antitumor and antiviral activities of 4-substituted 1,2,3-triazolyl-2,3-dibenzyl-L-ascorbic acid derivatives. European journal of medicinal chemistry\| PubMed ID: 31586832	2019
A unique class of lignin derivatives displays broad anti-HIV activity by interacting with the viral envelope. Virus research\| PubMed ID: 31618614	2019
Preprotein signature for full susceptibility to the co-translational translocation inhibitor cyclotriazadisulfonamide. Traffic (Copenhagen, Denmark)\| PubMed ID: 31675144	2020
Novel Isoxazolidine and γ-Lactam Analogues of Homonucleosides. Molecules (Basel, Switzerland)\| PubMed ID: 31698778	2019
Tryptophan Trimers and Tetramers Inhibit Dengue and Zika Virus Replication by Interfering with Viral Attachment Processes. Antimicrobial agents and chemotherapy\| PubMed ID: 31932383	2020
Design, synthesis and biological evaluation of 2-alkoxycarbonyl-3-anilinoindoles as a new class of potent inhibitors of tubulin polymerization. Bioorganic chemistry\| PubMed ID: 32086053	2020
A chimeric yellow fever-Zika virus vaccine candidate fully protects against yellow fever virus infection in mice. Emerging microbes & infections\| PubMed ID: 32116148	2020
Synthesis, antiviral, cytotoxic and cytostatic evaluation of -(phosphonoalkyl)uracil derivatives. Monatshefte fur chemie\| PubMed ID: 32214481	2016
Acyclic nucleoside phosphonates containing the amide bond: hydroxy derivatives. Monatshefte fur chemie\| PubMed ID: 32214483	2019
Synthesis of novel -acyl--d-glucopyranosylamines and ureas as potential lead cytostatic agents. Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents\| PubMed ID: 32214768	2016
Early protein expression profile in bronchoalveolar lavage fluid and clinical outcomes in primary graft dysfunction after lung transplantation. European journal of cardio-thoracic surgery : official journal of the European Association for Cardio-thoracic Surgery\| PubMed ID: 32267918	2020
Novel isoxazolidine analogues of homonucleosides and homonucleotides. Tetrahedron\| PubMed ID: 32287430	2016
Prodrugs of γ-Alkyl-Modified Nucleoside Triphosphates: Improved Inhibition of HIV Reverse Transcriptase. Angewandte Chemie (International ed. in English)\| PubMed ID: 32379948	2020
Anti-HIV-Active Nucleoside Triphosphate Prodrugs. Journal of medicinal chemistry\| PubMed ID: 32421343	2020
Lipophilic Triphosphate Prodrugs of Various Nucleoside Analogues. Journal of medicinal chemistry\| PubMed ID: 32515595	2020
Water-soluble fullerene-based nanostructures with promising antiviral and myogenic activity. Chemical communications (Cambridge, England)\| PubMed ID: 32748905	2020
Discovery of HIV entry inhibitors via a hybrid CXCR4 and CCR5 receptor pharmacophore-based virtual screening approach. European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences\| PubMed ID: 32890663	2020
Synthesis of new riboflavin modified ODNs: Effect of riboflavin moiety on the G-quadruplex arrangement and stability. Bioorganic chemistry\| PubMed ID: 32919132	2020
Membrane Permeable, Bioreversibly Modified Prodrugs of Nucleoside Diphosphate-γ-Phosphonates. Journal of medicinal chemistry\| PubMed ID: 32991174	2020
Itaconic acid hybrids as potential anticancer agents. Molecular diversity\| PubMed ID: 33043404	2022
Alkylated benzimidazoles: Design, synthesis, docking, DFT analysis, ADMET property, molecular dynamics and activity against HIV and YFV. Computational biology and chemistry\| PubMed ID: 33068917	2020
Thiophene-based water-soluble fullerene derivatives as highly potent antiherpetic pharmaceuticals. Organic & biomolecular chemistry\| PubMed ID: 33084716	2020
γ-Non-Symmetrically Dimasked TriPPPro Prodrugs as Potential Antiviral Agents against HIV. ChemMedChem\| PubMed ID: 33089929	2021
Development of a Novel SPR Assay to Study CXCR4-Ligand Interactions. Biosensors\| PubMed ID: 33096938	2020
γ-Ketobenzyl-Modified Nucleoside Triphosphate Prodrugs as Potential Antivirals. Journal of medicinal chemistry\| PubMed ID: 33186038	2020
STAT2 signaling restricts viral dissemination but drives severe pneumonia in SARS-CoV-2 infected hamsters. Nature communications\| PubMed ID: 33203860	2020
A single-dose live-attenuated YF17D-vectored SARS-CoV-2 vaccine candidate. Nature\| PubMed ID: 33260195	2021
Synthesis, Molecular Docking and Preliminary Antileukemic Activity of 4-Methoxybenzyl Derivatives Bearing Imidazo[2,1-b][1,3,4]thiadiazole. Chemistry & biodiversity\| PubMed ID: 33274824	2021
Characterization of the Carbohydrate-Binding Agents HHA, GNA, and UDA as Inhibitors of Influenza A and B Virus Replication. Antimicrobial agents and chemotherapy\| PubMed ID: 33288640	2021
Palladium-catalyzed cross-coupling reactions on a bromo-naphthalene scaffold in the search for novel human CC chemokine receptor 8 (CCR8) antagonists. Bioorganic chemistry\| PubMed ID: 33383325	2021
Discovery of 3-phenyl- and 3-N-piperidinyl-isothiazolo[4,3-b]pyridines as highly potent inhibitors of cyclin G-associated kinase. European journal of medicinal chemistry\| PubMed ID: 33497888	2021
A novel experimental porcine model to assess the impact of differential pulmonary blood flow on ischemia-reperfusion injury after unilateral lung transplantation. Intensive care medicine experimental\| PubMed ID: 33543363	2021
Synthesis, in silico ADME, molecular docking and in vitro cytotoxicity evaluation of stilbene linked 1,2,3-triazoles. Heliyon\| PubMed ID: 33553718	2021
FO-SPR biosensor calibrated with recombinant extracellular vesicles enables specific and sensitive detection directly in complex matrices. Journal of extracellular vesicles\| PubMed ID: 33664936	2021
Corrigendum to 'Discovery of HIV entry inhibitors via a hybrid CXCR4 and CCR5 receptor pharmacophore-based virtual screening approach' [European Journal of Pharmaceutical Sciences 155 (2020)... European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences\| PubMed ID: 33814256	2021
Biological characterization of ligands targeting the human CC chemokine receptor 8 (CCR8) reveals the biased signaling properties of small molecule agonists. Biochemical pharmacology\| PubMed ID: 33872569	2021
Small Molecule Cyclotriazadisulfonamide Abrogates the Upregulation of the Human Receptors CD4 and 4-1BB and Suppresses In Vitro Activation and Proliferation of T Lymphocytes. Frontiers in immunology\| PubMed ID: 33968048	2021
A Novel Series of Indole Alkaloid Derivatives Inhibit Dengue and Zika Virus Infection by Interference with the Viral Replication Complex. Antimicrobial agents and chemotherapy\| PubMed ID: 34001508	2021
Active Components from Prevent HIV-1 Entry by Distinct Mechanisms of Action. International journal of molecular sciences\| PubMed ID: 34068829	2021
Discovery of ( ±)-3-(1H-pyrazol-1-yl)-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4] thiadiazine derivatives with promising in vitro anticoronavirus and antitumoral activity. Molecular diversity\| PubMed ID: 34165689	2022
Broad spectrum anti-coronavirus activity of a series of anti-malaria quinoline analogues. Antiviral research\| PubMed ID: 34217752	2021
Labyrinthopeptin A1 inhibits dengue and Zika virus infection by interfering with the viral phospholipid membrane. Virology\| PubMed ID: 34274562	2021
Internal Disulfide Bonding and Glycosylation of Interleukin-7 Protect Against Proteolytic Inactivation by Neutrophil Metalloproteinases and Serine Proteases. Frontiers in immunology\| PubMed ID: 34276694	2021
Novel N-Substituted 3-Aryl-4-(diethoxyphosphoryl)azetidin-2-ones as Antibiotic Enhancers and Antiviral Agents in Search for a Successful Treatment of Complex Infections. International journal of molecular sciences\| PubMed ID: 34360797	2021
Exploring the dNTP -binding site of HIV-1 reverse transcriptase for inhibitor design. European journal of medicinal chemistry\| PubMed ID: 34425311	2021
Water-Promoted Reaction of CArCl Compounds with Thiophenes Delivers a Family of Multifunctional Fullerene Derivatives with Selective Antiviral Properties. Organic letters\| PubMed ID: 34468156	2021
A Proteomic Study on the Membrane Protein Fraction of T Cells Confirms High Substrate Selectivity for the ER Translocation Inhibitor Cyclotriazadisulfonamide. Molecular & cellular proteomics : MCP\| PubMed ID: 34481949	2021
D-Peptide-Based Probe for CXCR4-Targeted Molecular Imaging and Radionuclide Therapy. Pharmaceutics\| PubMed ID: 34683912	2021
Synthesis and Anti-HIV Activity of a Novel Series of Isoquinoline-Based CXCR4 Antagonists. Molecules (Basel, Switzerland)\| PubMed ID: 34684878	2021
Lung Microenvironments and Disease Progression in Fibrotic Hypersensitivity Pneumonitis. American journal of respiratory and critical care medicine\| PubMed ID: 34724391	2022
Atypical response to bacterial coinfection and persistent neutrophilic bronchoalveolar inflammation distinguish critical COVID-19 from influenza. JCI insight\| PubMed ID: 34793331	2022
Peripherally-driven myeloid NFkB and IFN/ISG responses predict malignancy risk, survival, and immunotherapy regime in ovarian cancer. Journal for immunotherapy of cancer\| PubMed ID: 34795003	2021
Skeleton binding protein-1-mediated parasite sequestration inhibits spontaneous resolution of malaria-associated acute respiratory distress syndrome. PLoS pathogens\| PubMed ID: 34843584	2021
Sliding of HIV-1 reverse transcriptase over DNA creates a transient P pocket - targeting P-pocket by fragment screening. Nature communications\| PubMed ID: 34880240	2021
Deciphering the Role of Extracellular Vesicles Derived from ZIKV-Infected hcMEC/D3 Cells on the Blood-Brain Barrier System. Viruses\| PubMed ID: 34960632	2021
Anthranilamides with quinoline and β-carboline scaffolds: design, synthesis, and biological activity. Molecular diversity\| PubMed ID: 34997441	2022
Synthesis, in vitro cytotoxicity, molecular docking and ADME study of some indolin-2-one linked 1,2,3-triazole derivatives. Computational biology and chemistry\| PubMed ID: 35168158	2022
Targeting chemokine receptors from the inside-out: discovery and development of small-molecule intracellular antagonists. Chemical communications (Cambridge, England)\| PubMed ID: 35274633	2022
Circulating Donor-Specific Anti-HLA Antibodies Associate With Immune Activation Independent of Kidney Transplant Histopathological Findings. Frontiers in immunology\| PubMed ID: 35281018	2022
Identification of novel chemotypes as CXCR2 antagonists via a scaffold hopping approach from a thiazolo[4,5-d]pyrimidine. European journal of medicinal chemistry\| PubMed ID: 35313168	2022
A Set of Experimentally Validated Decoys for the Human CC Chemokine Receptor 7 (CCR7) Obtained by Virtual Screening. Frontiers in pharmacology\| PubMed ID: 35370691	2022
Innate Lymphoid Cells Are Required to Induce Airway Hyperreactivity in a Murine Neutrophilic Asthma Model. Frontiers in immunology\| PubMed ID: 35371094	2022
In silico design, synthesis and anti-HIV activity of quinoline derivatives as non-nucleoside reverse transcriptase inhibitors (NNRTIs). Computational biology and chemistry\| PubMed ID: 35395595	2022
Effect of Particle Carriers for Intraperitoneal Drug Delivery on the Course of Ovarian Cancer and Its Immune Microenvironment in a Mouse Model. Pharmaceutics\| PubMed ID: 35456521	2022
Stimulation of the atypical chemokine receptor 3 (ACKR3) by a small-molecule agonist attenuates fibrosis in a preclinical liver but not lung injury model. Cellular and molecular life sciences : CMLS\| PubMed ID: 35562519	2022
Discovery of 2-Phenylquinolines with Broad-Spectrum Anti-coronavirus Activity. ACS medicinal chemistry letters\| PubMed ID: 35571875	2022
The discovery of Zika virus NS2B-NS3 inhibitors with antiviral activity via an integrated virtual screening approach. European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences\| PubMed ID: 35618201	2022
SARS-CoV-2 Virion Infectivity and Cytokine Production in Primary Human Airway Epithelial Cells. Viruses\| PubMed ID: 35632693	2022
Potent neutralizing anti-SARS-CoV-2 human antibodies cure infection with SARS-CoV-2 variants in hamster model. iScience\| PubMed ID: 35813873	2022
Cryo-EM structures of wild-type and E138K/M184I mutant HIV-1 RT/DNA complexed with inhibitors doravirine and rilpivirine. Proceedings of the National Academy of Sciences of the United States of America\| PubMed ID: 35858448	2022
Cellular Electrical Impedance as a Method to Decipher CCR7 Signalling and Biased Agonism. International journal of molecular sciences\| PubMed ID: 36012168	2022
Triphosphate Prodrugs of the Anti-HIV-Active Compound 3'-Deoxy-3'-fluorothymidine (FLT). Journal of medicinal chemistry\| PubMed ID: 36099330	2022
Carbohydrate-binding protein from stinging nettle as fusion inhibitor for SARS-CoV-2 variants of concern. Frontiers in cellular and infection microbiology\| PubMed ID: 36111239	2022
Corrigendum: Innate lymphoid cells are required to induce airway hyperreactivity in a murine neutrophilic asthma model. Frontiers in immunology\| PubMed ID: 36211405	2022
Can we attenuate ischaemia-reperfusion injury of allografts in a porcine left lung transplant models by adsorption of cytokines? European journal of cardio-thoracic surgery : official journal of the European Association for Cardio-thoracic Surgery\| PubMed ID: 36214633	2022
Design, Synthesis, Anti-Varicella-Zoster and Antimicrobial Activity of (Isoxazolidin-3-yl)Phosphonate Conjugates of N1-Functionalised Quinazoline-2,4-Diones. Molecules (Basel, Switzerland)\| PubMed ID: 36235061	2022
A stabilized CXCL9(74-103)-derived peptide selectively inhibits proliferation, adhesion and metastasis of tumor cells that express high levels of heparan sulfate. International journal of biological macromolecules\| PubMed ID: 36272565	2022
Synthesis and evaluation of 3-alkynyl-5-aryl-7-aza-indoles as broad-spectrum antiviral agents. Frontiers in chemistry\| PubMed ID: 36385995	2022
Development of a live biotherapeutic throat spray with lactobacilli targeting respiratory viral infections. Microbial biotechnology\| PubMed ID: 36468246	2023
Systemic cytokines and GlycA discriminate disease status and predict corticosteroid response in HTLV-1-associated neuroinflammation. Journal of neuroinflammation\| PubMed ID: 36482436	2022
Design and synthesis of a new series of hybrids of functionalised N-[(1H-1,2,3-triazol-4-yl)methyl]quinazoline-2,4-dione with antiviral activity against Respiratory Syncytial Virus. Antiviral research\| PubMed ID: 36587900	2023
Identification of Polyphenol Derivatives as Novel SARS-CoV-2 and DENV Non-Nucleoside RdRp Inhibitors. Molecules (Basel, Switzerland)\| PubMed ID: 36615354	2022
FLUIDOT: A Modular Microfluidic Platform for Single-Cell Study and Retrieval, with Applications in Drug Tolerance Screening and Antibody Mining. Small methods\| PubMed ID: 36642827	2023
Visible-Light-Promoted Tandem Thiol-Ene Click Reaction/Transannular Cyclization and Regioselective Cyclopropane Ring-Opening to Construct Sulfur-Containing Diterpenes. Organic letters\| PubMed ID: 36662155	2023
Exploration of Pyrido[3,4-]pyrimidines as Antagonists of the Human Chemokine Receptor CXCR2. Molecules (Basel, Switzerland)\| PubMed ID: 36903345	2023
A regioselective step-by-step CCl functionalization approach affords a novel family of CArTh'Th''H fullerene derivatives with promising antiviral properties. Chemical communications (Cambridge, England)\| PubMed ID: 36916636	2023
Optimization of triazolo[4,5-d]pyrimidines towards human CC chemokine receptor 7 (CCR7) antagonists. European journal of medicinal chemistry\| PubMed ID: 36924670	2023