Véronique Gouverneur

Publications

• Organophotoredox Hydrodefluorination of Trifluoromethylarenes with Translational Applicability to Drug Discovery
  Journal of the American Chemical Society. May, 2020  |   Pubmed ID: 32379965
• [F]AZD2461, an Insight on Difference in PARP Binding Profiles for DNA Damage Response PET Imaging
  Molecular Imaging and Biology. Apr, 2020  |   Pubmed ID: 32342268
• Hydrosulfonylation of Alkenes with Sulfonyl Chlorides Under Visible Light Activation
  Angewandte Chemie (International Ed. in English). Jul, 2020  |   Pubmed ID: 32286720
• Manual and Automated Cu-mediated Radiosynthesis of the PARP Inhibitor [F]olaparib
  Nature Protocols. 04, 2020  |   Pubmed ID: 32111986
• F-Trifluoromethanesulfinate Enables Direct C-H F-Trifluoromethylation of Native Aromatic Residues in Peptides
  Journal of the American Chemical Society. 01, 2020  |   Pubmed ID: 31913613
• Silyl Radical-Mediated Activation of Sulfamoyl Chlorides Enables Direct Access to Aliphatic Sulfonamides from Alkenes
  Journal of the American Chemical Society. 01, 2020  |   Pubmed ID: 31881153
• Imaging of Translocator Protein Upregulation is Selective for Pro-inflammatory Polarized Astrocytes and Microglia
  Glia. 02, 2020  |   Pubmed ID: 31479168
• Hydrodifluoromethylation of Alkenes with Difluoroacetic Acid
  Angewandte Chemie (International Ed. in English). 06, 2019  |   Pubmed ID: 31020767
• Synthesis of F-difluoromethylarenes Using Aryl Boronic Acids, Ethyl Bromofluoroacetate and [F]fluoride
  Chemical Science. Mar, 2019  |   Pubmed ID: 30996907
• Hydrogen Bonding Phase-Transfer Catalysis with Potassium Fluoride: Enantioselective Synthesis of β-Fluoroamines
  Journal of the American Chemical Society. 02, 2019  |   Pubmed ID: 30689372
• Synthesis and Reactivity of α-Cumyl Bromodifluoromethanesulfenate: Application to the Radiosynthesis of [ F]ArylSCF
  Angewandte Chemie (International Ed. in English). Feb, 2019  |   Pubmed ID: 30575245
• PET Imaging of PARP Expression Using F-Olaparib
  Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. 04, 2019  |   Pubmed ID: 30389822
• Boron Reagents for Divergent Radiochemistry
  Chemical Society Reviews. Sep, 2018  |   Pubmed ID: 30140795
• Asymmetric Nucleophilic Fluorination Under Hydrogen Bonding Phase-transfer Catalysis
  Science (New York, N.Y.). 05, 2018  |   Pubmed ID: 29748281
• Controlled Single and Double Iodofluorination of Alkynes with DIH- and HF-Based Reagents
  Organic Letters. 03, 2018  |   Pubmed ID: 29493242
• Highly Diastereoselective Synthesis of Trifluoromethyl Indolines by Interceptive Benzylic Decarboxylative Cycloaddition of Nonvinyl, Trifluoromethyl Benzoxazinanones with Sulfur Ylides Under Palladium Catalysis
  Organic Letters. 03, 2018  |   Pubmed ID: 29474077
• Selective Radical Trifluoromethylation of Native Residues in Proteins
  Journal of the American Chemical Society. 02, 2018  |   Pubmed ID: 29301396
• F-Trifluoromethylation of Unmodified Peptides with 5-F-(Trifluoromethyl)dibenzothiophenium Trifluoromethanesulfonate
  Journal of the American Chemical Society. 02, 2018  |   Pubmed ID: 29301394
• Derisking the Cu-Mediated F-Fluorination of Heterocyclic Positron Emission Tomography Radioligands
  Journal of the American Chemical Society. 06, 2017  |   Pubmed ID: 28548849
• The Dual Role of Thiourea in the Thiotrifluoromethylation of Alkenes
  Chemical Science. Feb, 2017  |   Pubmed ID: 28451260
• Synthesis and Reactivity of F-Labeled α,α-Difluoro-α-(aryloxy)acetic Acids
  Organic Letters. 02, 2017  |   Pubmed ID: 28085289
• Twisting the Ethano-Tröger's Base: the Bisamide
  Organic & Biomolecular Chemistry. Jan, 2017  |   Pubmed ID: 27966723
• Targeting Telomerase with Radiolabeled Inhibitors
  European Journal of Medicinal Chemistry. Jan, 2017  |   Pubmed ID: 27657809
• Asymmetric F-fluorination for Applications in Positron Emission Tomography
  Chemical Science. Mar, 2016  |   Pubmed ID: 28808536
• Bridging the Gaps in F PET Tracer Development
  Nature Chemistry. 12, 2016  |   Pubmed ID: 27995923
• Radiosynthesis of SPECT Tracers Via a Copper Mediated I Iodination of (hetero)aryl Boron Reagents
  Chemical Communications (Cambridge, England). Nov, 2016  |   Pubmed ID: 27775106
• Hydrogen-Bonded Homoleptic Fluoride-Diarylurea Complexes: Structure, Reactivity, and Coordinating Power
  Journal of the American Chemical Society. Oct, 2016  |   Pubmed ID: 27608274
• Ultrafast Click Chemistry with Fluorosydnones
  Angewandte Chemie (International Ed. in English). 09, 2016  |   Pubmed ID: 27560312
• Enhanced Copper-mediated (18)F-fluorination of Aryl Boronic Esters Provides Eight Radiotracers for PET Applications
  Chemical Communications (Cambridge, England). Jun, 2016  |   Pubmed ID: 27241832
• Copper-Catalyzed Insertion into Heteroatom-Hydrogen Bonds with Trifluorodiazoalkanes
  Angewandte Chemie (International Ed. in English). Mar, 2016  |   Pubmed ID: 26880039
• (18)F-Labeling of Arenes and Heteroarenes for Applications in Positron Emission Tomography
  Chemical Reviews. Jan, 2016  |   Pubmed ID: 26751274
• Synthesis and Characterization of a Novel N-F Reagent Derived from the Ethano-Tröger's Base: (1)J(FN) Coupling Constants As a Signature for the N-F Bond
  Chemical Communications (Cambridge, England). Jan, 2016  |   Pubmed ID: 26658721
• Coordination Diversity in Hydrogen-bonded Homoleptic Fluoride-alcohol Complexes Modulates Reactivity
  Chemical Science. Sep, 2015  |   Pubmed ID: 29449931
• Synthesis of F-Arenes from Spirocyclic Iodonium(III) Ylides Via Continuous-Flow Microfluidics
  Journal of Fluorine Chemistry. Oct, 2015  |   Pubmed ID: 27512233
• Organomediated Enantioselective (18)F Fluorination for PET Applications
  Angewandte Chemie (International Ed. in English). Nov, 2015  |   Pubmed ID: 26360631
• (18)F-Labeling of Aryl-SCF3, -OCF3 and -OCHF2 with [(18)F]Fluoride
  Angewandte Chemie (International Ed. in English). Aug, 2015  |   Pubmed ID: 26140357
• Cross-Coupling of [2-Aryl-1,1,2,2-tetrafluoroethyl](trimethyl)silanes with Aryl Halides
  Organic Letters. Jul, 2015  |   Pubmed ID: 26126930
• Recruitment and Immobilization of a Fluorinated Biomarker Across an Interfacial Phospholipid Film Using a Fluorocarbon Gas
  Angewandte Chemie (International Ed. in English). Jul, 2015  |   Pubmed ID: 26068966
• A Dual Radiolabelling Approach for Tracking Metal Complexes: Investigating the Speciation of Copper Bis(thiosemicarbazonates) in Vitro and in Vivo
  Metallomics : Integrated Biometal Science. May, 2015  |   Pubmed ID: 25768310
• Anti-CD20 Inhibits T Cell-mediated Pathology and Microgliosis in the Rat Brain
  Annals of Clinical and Translational Neurology. Sep, 2014  |   Pubmed ID: 25493280
• Asymmetric Fluorocyclizations of Alkenes
  Accounts of Chemical Research. Dec, 2014  |   Pubmed ID: 25379791
• Diversity-oriented Approach to CF3CHF-, CF3CFBr-, CF3CF2-, (CF3)2CH-, and CF3(SCF3)CH-substituted Arenes from 1-(diazo-2,2,2-trifluoroethyl)arenes
  Organic Letters. Nov, 2014  |   Pubmed ID: 25379614
• A General Copper-mediated Nucleophilic 18F fluorination of Arenes
  Angewandte Chemie (International Ed. in English). Jul, 2014  |   Pubmed ID: 24916101
• Cis-Specific Hydrofluorination of Alkenylarenes Under Palladium Catalysis Through an Ionic Pathway
  Angewandte Chemie (International Ed. in English). Apr, 2014  |   Pubmed ID: 24644083
• Glial Activation in the Early Stages of Brain Metastasis: TSPO As a Diagnostic Biomarker
  Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. Feb, 2014  |   Pubmed ID: 24434290
• A Comparison of the Behavior of (64)Cu-acetate and (64)Cu-ATSM in Vitro and in Vivo
  Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. Jan, 2014  |   Pubmed ID: 24337603
• Enhanced Aqueous Suzuki-Miyaura Coupling Allows Site-specific Polypeptide 18F-labeling
  Journal of the American Chemical Society. Sep, 2013  |   Pubmed ID: 23991754
• Intramolecular OH···FC Hydrogen Bonding in Fluorinated Carbohydrates: CHF is a Better Hydrogen Bond Acceptor Than CF2
  Angewandte Chemie (International Ed. in English). Sep, 2013  |   Pubmed ID: 23960019
• Asymmetric Electrophilic Fluorocyclization with Carbon Nucleophiles
  Angewandte Chemie (International Ed. in English). Sep, 2013  |   Pubmed ID: 23873744
• Catalytic Decarboxylative Fluorination for the Synthesis of Tri- and Difluoromethyl Arenes
  Organic Letters. Jun, 2013  |   Pubmed ID: 23687958
• Trifluoromethylation of Allylsilanes Under Photoredox Catalysis
  Organic Letters. Mar, 2013  |   Pubmed ID: 23465076
• Catalytic Hydrotrifluoromethylation of Unactivated Alkenes
  Journal of the American Chemical Society. Feb, 2013  |   Pubmed ID: 23373772
• [18F]fluorination of an Arylboronic Ester Using [18F]selectfluor Bis(triflate): Application to 6-[18F]fluoro-L-DOPA
  Chemical Communications (Cambridge, England). Feb, 2013  |   Pubmed ID: 23321570
• 18F Labeling of Arenes
  Angewandte Chemie (International Ed. in English). Nov, 2012  |   Pubmed ID: 23086547
• Conformational Analysis of Fluorinated Pyrrolidines Using 19F-1H Scalar Couplings and Heteronuclear NOEs
  Chemistry (Weinheim an Der Bergstrasse, Germany). Oct, 2012  |   Pubmed ID: 22991298
• Synthesis of 3-fluoropyrrolidines and 4-fluoropyrrolidin-2-ones from Allylic Fluorides
  Chemistry (Weinheim an Der Bergstrasse, Germany). Oct, 2012  |   Pubmed ID: 22991281
• Trifluoromethylation of Allylsilanes Under Copper Catalysis
  Chemistry (Weinheim an Der Bergstrasse, Germany). Jul, 2012  |   Pubmed ID: 22692972
• Metal-free Oxidative Fluorination of Phenols with [18F]fluoride
  Angewandte Chemie (International Ed. in English). Jul, 2012  |   Pubmed ID: 22639017
• Palladium-catalyzed Substitution and Cross-coupling of Benzylic Fluorides
  Organic Letters. Jun, 2012  |   Pubmed ID: 22594918
• Transition Metal Catalysis and Nucleophilic Fluorination
  Chemical Communications (Cambridge, England). Mar, 2012  |   Pubmed ID: 22334339
• A Fluorous and Click Approach for Screening Potential PET Probes: Evaluation of Potential Hypoxia Biomarkers
  Bioorganic & Medicinal Chemistry. Jan, 2012  |   Pubmed ID: 22130421
• Hypoxia Imaging Using PET and SPECT: the Effects of Anesthetic and Carrier Gas on [Cu]-ATSM, [Tc]-HL91 and [F]-FMISO Tumor Hypoxia Accumulation
  PloS One. 2011  |   Pubmed ID: 22102855
• Organocatalyzed Enantioselective Fluorocyclizations
  Angewandte Chemie (International Ed. in English). Aug, 2011  |   Pubmed ID: 21751319
• Au(I) /Au(III) Catalysis: an Alternative Approach for C-C Oxidative Coupling
  Chemistry (Weinheim an Der Bergstrasse, Germany). Jul, 2011  |   Pubmed ID: 21678513
• Palladium-catalyzed Allylic Fluorination
  Angewandte Chemie (International Ed. in English). Mar, 2011  |   Pubmed ID: 21370349
• The Chemoselective One-step Alkylation and Isolation of Thiophosphorylated Cdk2 Substrates in the Presence of Native Cysteine
  Chembiochem : a European Journal of Chemical Biology. Mar, 2011  |   Pubmed ID: 21305681
• The Traceless Staudinger Ligation for Indirect 18F-radiolabelling
  Organic & Biomolecular Chemistry. Jan, 2011  |   Pubmed ID: 21103523
• Gold-catalyzed Cascade Cyclization-oxidative Alkynylation of Allenoates
  Organic Letters. Nov, 2010  |   Pubmed ID: 20936849
• Catalytic Enantioselective Synthesis of P-stereogenic Compounds
  Chemical Communications (Cambridge, England). Oct, 2010  |   Pubmed ID: 20835471
• Radiosynthesis and Evaluation of [18F]Selectfluor Bis(triflate)
  Angewandte Chemie (International Ed. in English). Sep, 2010  |   Pubmed ID: 20715033
• Pre-clinical Evaluation of a 3-nitro-1,2,4-triazole Analogue of [18F]FMISO As Hypoxia-selective Tracer for PET
  Nuclear Medicine and Biology. Jul, 2010  |   Pubmed ID: 20610161
• Orthogonal 18F and 64Cu Labelling of Functionalised Bis(thiosemicarbazonato) Complexes
  Chemical Communications (Cambridge, England). Jun, 2010  |   Pubmed ID: 20407674
• Bis(thiosemicarbazones) As Bifunctional Chelators for the Room Temperature 64-copper Labeling of Peptides
  Dalton Transactions (Cambridge, England : 2003). Apr, 2010  |   Pubmed ID: 20354615
• Gold-catalyzed Intramolecular Oxidative Cross-coupling of Nonactivated Arenes
  Chemistry (Weinheim an Der Bergstrasse, Germany). Apr, 2010  |   Pubmed ID: 20340120
• Synthesis and O-phosphorylation of 3,3,4,4-tetrafluoroaryl-C-nucleoside Analogues
  Organic & Biomolecular Chemistry. Mar, 2010  |   Pubmed ID: 20204220
• Diastereoselective Synthesis of P-stereogenic Heterocycles Via Enyne Ring-closing Metathesis
  Organic Letters. Mar, 2010  |   Pubmed ID: 20184294
• Developments in Fluorocyclization Methodologies
  Future Medicinal Chemistry. Aug, 2009  |   Pubmed ID: 21426084
• Transition-metal-mediated Reactions for C(sp2)-F Bond Construction: the State of Play
  Angewandte Chemie (International Ed. in English). 2009  |   Pubmed ID: 19827068
• Chemistry. A New Departure in Fluorination Chemistry
  Science (New York, N.Y.). Sep, 2009  |   Pubmed ID: 19779178
• Electrophilic Fluorocyclization of Allyl Silanes
  Angewandte Chemie (International Ed. in English). 2009  |   Pubmed ID: 19697388
• Synthesis and Reactivity of Novel Gamma-phosphate Modified ATP Analogues
  Bioorganic & Medicinal Chemistry Letters. Jul, 2009  |   Pubmed ID: 19410453
• Diels-Alder Exo Selectivity in Terminal-substituted Dienes and Dienophiles: Experimental Discoveries and Computational Explanations
  Journal of the American Chemical Society. Feb, 2009  |   Pubmed ID: 19154113
• Enantioselective Synthesis of P-stereogenic Phosphinates and Phosphine Oxides by Molybdenum-catalyzed Asymmetric Ring-closing Metathesis
  Angewandte Chemie (International Ed. in English). 2009  |   Pubmed ID: 19101976
• A Two-directional Approach to Enantiopure 1,4-difluoro-cyclohexenes: Synthesis of Difluorinated Cyclitol Analogues
  Organic Letters. Oct, 2008  |   Pubmed ID: 18763795
• Gold(I)-catalyzed Alkoxyhalogenation of Beta-hydroxy-alpha,alpha-difluoroynones
  Angewandte Chemie (International Ed. in English). 2008  |   Pubmed ID: 18683842
• Fluorous Synthesis of Allylic Fluorides: C-F Bond Formation As the Detagging Process
  Chemical Communications (Cambridge, England). Aug, 2008  |   Pubmed ID: 18665278
• The Chemistry of Propargylic and Allylic Fluorides
  Chemical Reviews. Jun, 2008  |   Pubmed ID: 18543877
• Stereospecific Anti SE2' Fluorination of Allenylsilanes: Synthesis of Enantioenriched Propargylic Fluorides
  Organic & Biomolecular Chemistry. May, 2008  |   Pubmed ID: 18452005
• Fluorine-directed Diastereoselective Iodocyclizations
  Angewandte Chemie (International Ed. in English). 2008  |   Pubmed ID: 18022878
• Single and Double Stereoselective Fluorination of (E)-allylsilanes
  Beilstein Journal of Organic Chemistry. Oct, 2007  |   Pubmed ID: 17961218
• Synthesis and Reactivity of [18F]-N-fluorobenzenesulfonimide
  Chemical Communications (Cambridge, England). Jun, 2007  |   Pubmed ID: 17844736
• A Concise Synthesis of Enantioenriched Fluorinated Carbocycles
  Angewandte Chemie (International Ed. in English). 2007  |   Pubmed ID: 17549786
• Enantioselective Organocatalytic Aldol Reaction of Ynones and Its Synthetic Applications
  Organic Letters. Nov, 2006  |   Pubmed ID: 17078732
• Sequential Desymmetrization-fluorination: Enantioselective Synthesis of Fluorinated Cyclitols
  Chemistry (Weinheim an Der Bergstrasse, Germany). Dec, 2006  |   Pubmed ID: 17066392
• Pd(II)-catalyzed Cascade Wacker-Heck Reaction: Chemoselective Coupling of Two Electron-deficient Reactants
  The Journal of Organic Chemistry. Oct, 2006  |   Pubmed ID: 17064010
• Synthesis of Propargylic Fluorides from Allenylsilanes
  Chemical Communications (Cambridge, England). Oct, 2006  |   Pubmed ID: 17024266
• Intramolecular Hetero-Michael Addition of Beta-hydroxyenones for the Preparation of Highly Substituted Tetrahydropyranones
  Chemistry (Weinheim an Der Bergstrasse, Germany). Sep, 2006  |   Pubmed ID: 16819725
• Enantioselective Synthesis of a Key "A-ring" Intermediate for the Preparation of 1alpha-fluoro Vitamin D3 Analogues
  The Journal of Organic Chemistry. Jul, 2006  |   Pubmed ID: 16808527
• Catalytic Asymmetric Fluorinations
  Organic & Biomolecular Chemistry. Jun, 2006  |   Pubmed ID: 16729117
• Electrophilic Fluorination of Organosilanes
  Organic & Biomolecular Chemistry. Jan, 2006  |   Pubmed ID: 16357989
• Diastereoselective Ring-closing Metathesis: Synthesis of P-stereogenic Phosphinates from Prochiral Phosphinic Acid Derivatives
  The Journal of Organic Chemistry. Dec, 2005  |   Pubmed ID: 16356003
• Palladium-catalyzed Oxidative Cyclizations: Synthesis of Dihydropyranones and Furanones
  The Journal of Organic Chemistry. Oct, 2005  |   Pubmed ID: 16209595
• Synthesis of Novel Enantiopure Fluorinated Building Blocks from Acyclic Chiral Allylsilanes
  Organic Letters. Sep, 2005  |   Pubmed ID: 16178567
• Biocatalytic Approaches to Hetero-Diels-Alder Adducts of Carbonyl Compounds
  Chemistry (Weinheim an Der Bergstrasse, Germany). Oct, 2005  |   Pubmed ID: 16003810
• Electrophilic Fluorodesilylation of Allenylmethylsilanes: a Novel Entry to 2-fluoro-1,3-dienes
  Organic Letters. Mar, 2005  |   Pubmed ID: 15787483
• A Catalytic Asymmetric Bioorganic Route to Enantioenriched Tetrahydro- and Dihydropyranones
  Journal of the American Chemical Society. Feb, 2005  |   Pubmed ID: 15686381
• Stereoselective Synthesis of Internal Allylic Fluorides
  Organic & Biomolecular Chemistry. Apr, 2004  |   Pubmed ID: 15064784
• Oxidative Cyclization of Beta-hydroxyenones with Palladium(II): a Novel Entry to 2,3-dihydro-4H-pyran-4-ones
  Organic Letters. Jan, 2004  |   Pubmed ID: 14703358
• Sequential Cross-metathesis/electrophilic Fluorodesilylation: a Novel Entry to Functionalized Allylic Fluorides
  Organic Letters. Dec, 2003  |   Pubmed ID: 14653700
• Synthesis of Unprotected and Borane-protected Cyclic Phosphines Using Ru- and Mo- Based Olefin Metathesis Catalysts
  Organic & Biomolecular Chemistry. Nov, 2003  |   Pubmed ID: 14649914
• Regio- and Enantioselective Synthesis of Allylic Fluorides by Electrophilic Fluorodesilylation of Allyl Silanes
  Angewandte Chemie (International Ed. in English). Jul, 2003  |   Pubmed ID: 12876747
• Unprecedented Regiocontrol Using an Aldolase I Antibody
  Angewandte Chemie (International Ed. in English). Mar, 2002  |   Pubmed ID: 12491296
• Synthetic Applications of Electrophilic Fluorodesilylation
  Chemistry (Weinheim an Der Bergstrasse, Germany). Feb, 2002  |   Pubmed ID: 11857690