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Chapters
- 00:05Title
- 01:23General Thallium Flux Assay Procedure
- 05:04Checkerboard Analysis
- 07:22Results: High-throughput Screening for Small-molecule Modulators of Inward Rectifier Potassium Channels
- 09:27Conclusion
Tags
High-throughput ScreeningSmall-molecule ModulatorsInward Rectifier Potassium ChannelsDrug TargetsPharmacological ToolsMolecular PharmacologyS4 SuperfamilyVoltage-gated Potassium ChannelsPeptide Toxin ModulatorsBee Venom Toxin TertiapinKir1.1Kir3 ChannelsAntigenic PropertiesPoor BioavailabilityMetabolic StabilitySmall-molecule ProbesPhysiologyTherapeutic Potential
